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Pharmacological evaluation and molecular docking of new di-tert-butylphenol compound, LQFM-091, a new dual 5-LOX/COX inhibitor.
Lino, Roberta Campos; da Silva, Daiany Priscila Bueno; Florentino, Iziara Ferreira; da Silva, Dayane Moreira; Martins, José Luís Rodrigues; Batista, Daniel da Costa; Leite, Karla Carneiro de Siqueira; Villavicencio, Bianca; Vasconcelos, Géssica A; Silva, Andreia Luiza Pereira; de Ávila, Renato Ivan; Verli, Hugo; Valadares, Marize Campos; Gil, Eric de Souza; Vaz, Boniek G; Lião, Luciano M; Menegatti, Ricardo; Costa, Elson Alves.
Afiliação
  • Lino RC; Post-Graduate Program in Pharmaceutical Innovation, Faculty of Pharmacy, Federal University of Goiás, Goiânia, GO, Brazil.
  • da Silva DPB; Post-Graduate Program in Biological Sciences, Institute of Biological Sciences, Federal University of Goiás, Campus Samambaia, Goiânia, GO, Brazil.
  • Florentino IF; Post-Graduate Program in Biological Sciences, Institute of Biological Sciences, Federal University of Goiás, Campus Samambaia, Goiânia, GO, Brazil.
  • da Silva DM; Post-Graduate Program in Biological Sciences, Institute of Biological Sciences, Federal University of Goiás, Campus Samambaia, Goiânia, GO, Brazil.
  • Martins JLR; Post-Graduate Program in Biological Sciences, Institute of Biological Sciences, Federal University of Goiás, Campus Samambaia, Goiânia, GO, Brazil.
  • Batista DDC; Post-Graduate Program in Biological Sciences, Institute of Biological Sciences, Federal University of Goiás, Campus Samambaia, Goiânia, GO, Brazil.
  • Leite KCS; Laboratory of Medicinal Pharmaceutical Chemistry, Faculty of Pharmacy, Federal University of Goiás, Goiânia, GO, Brazil.
  • Villavicencio B; Center of Biotechnology, Federal University of Rio Grande do Sul, RS, Brazil.
  • Vasconcelos GA; Chemistry Institute, Laboratory of Chromatography and Mass Spectrometry, Federal University of Goiás, Goiânia, GO, Brazil.
  • Silva ALP; Laboratory of Pharmacology and Cell Toxicology, Faculty of Pharmacy, Federal University of Goiás, Goiânia, GO, Brazil.
  • de Ávila RI; Laboratory of Pharmacology and Cell Toxicology, Faculty of Pharmacy, Federal University of Goiás, Goiânia, GO, Brazil.
  • Verli H; Center of Biotechnology, Federal University of Rio Grande do Sul, RS, Brazil.
  • Valadares MC; Laboratory of Pharmacology and Cell Toxicology, Faculty of Pharmacy, Federal University of Goiás, Goiânia, GO, Brazil.
  • Gil ES; Laboratory of Medicinal Pharmaceutical Chemistry, Faculty of Pharmacy, Federal University of Goiás, Goiânia, GO, Brazil.
  • Vaz BG; Chemistry Institute, Laboratory of Chromatography and Mass Spectrometry, Federal University of Goiás, Goiânia, GO, Brazil.
  • Lião LM; Chemistry Institute, Federal University of Goias, Campus Samambaia, Goiânia, GO, Brazil.
  • Menegatti R; Laboratory of Medicinal Pharmaceutical Chemistry, Faculty of Pharmacy, Federal University of Goiás, Goiânia, GO, Brazil.
  • Costa EA; Department of Pharmacology, Institute of Biological Sciences, Federal University of Goiás, Campus Samambaia, Goiânia, GO, Brazil. Electronic address: xico@ufg.br.
Eur J Pharm Sci ; 106: 231-243, 2017 Aug 30.
Article em En | MEDLINE | ID: mdl-28599988

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fenóis / Inibidores de Lipoxigenase / Inibidores de Ciclo-Oxigenase Limite: Animals Idioma: En Revista: Eur J Pharm Sci Assunto da revista: FARMACIA / FARMACOLOGIA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Brasil País de publicação: Holanda

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fenóis / Inibidores de Lipoxigenase / Inibidores de Ciclo-Oxigenase Limite: Animals Idioma: En Revista: Eur J Pharm Sci Assunto da revista: FARMACIA / FARMACOLOGIA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Brasil País de publicação: Holanda