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Discovery of a highly potent and orally available importin-ß1 inhibitor that overcomes enzalutamide-resistance in advanced prostate cancer.
Huang, Jia-Luo; Yan, Xue-Long; Huang, Dong; Gan, Lu; Gao, Huahua; Fan, Run-Zhu; Li, Shen; Yuan, Fang-Yu; Zhu, Xinying; Tang, Gui-Hua; Chen, Hong-Wu; Wang, Junjian; Yin, Sheng.
Afiliación
  • Huang JL; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Yan XL; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Huang D; School of Pharmacy, Guizhou Medical University, Guian New District, Guizhou 550025, China.
  • Gan L; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Gao H; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Fan RZ; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Li S; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Yuan FY; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Zhu X; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Tang GH; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Chen HW; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
  • Wang J; School of Medicine, University of California Davis, Sacramento, CA 95817, USA.
  • Yin S; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, China.
Acta Pharm Sin B ; 13(12): 4934-4944, 2023 Dec.
Article en En | MEDLINE | ID: mdl-38045040

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: Acta Pharm Sin B Año: 2023 Tipo del documento: Article País de afiliación: China Pais de publicación: Países Bajos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: Acta Pharm Sin B Año: 2023 Tipo del documento: Article País de afiliación: China Pais de publicación: Países Bajos