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Discovery of Potent Pyrazoline-Based Covalent SARS-CoV-2 Main Protease Inhibitors.
Moon, Patrick; Zammit, Charlotte M; Shao, Qian; Dovala, Dustin; Boike, Lydia; Henning, Nathaniel J; Knapp, Mark; Spradlin, Jessica N; Ward, Carl C; Wolleb, Helene; Fuller, Daniel; Blake, Gabrielle; Murphy, Jason P; Wang, Feng; Lu, Yipin; Moquin, Stephanie A; Tandeske, Laura; Hesse, Matthew J; McKenna, Jeffrey M; Tallarico, John A; Schirle, Markus; Toste, F Dean; Nomura, Daniel K.
Afiliación
  • Moon P; Department of Chemistry, University of California, Berkeley, Berkeley, CA-94720, USA.
  • Zammit CM; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Shao Q; Department of Chemistry, University of California, Berkeley, Berkeley, CA-94720, USA.
  • Dovala D; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Boike L; Department of Chemistry, University of California, Berkeley, Berkeley, CA-94720, USA.
  • Henning NJ; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Knapp M; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Spradlin JN; Novartis Institutes for BioMedical Research, Emeryville, CA 94608, USA.
  • Ward CC; Department of Chemistry, University of California, Berkeley, Berkeley, CA-94720, USA.
  • Wolleb H; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Fuller D; Department of Chemistry, University of California, Berkeley, Berkeley, CA-94720, USA.
  • Blake G; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Murphy JP; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Wang F; Novartis Institutes for BioMedical Research, Emeryville, CA 94608, USA.
  • Lu Y; Department of Chemistry, University of California, Berkeley, Berkeley, CA-94720, USA.
  • Moquin SA; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Tandeske L; Department of Chemistry, University of California, Berkeley, Berkeley, CA-94720, USA.
  • Hesse MJ; Department of Molecular and Cell Biology, University of California, Berkeley, Berkeley, CA-94720, USA.
  • McKenna JM; Department of Chemistry, University of California, Berkeley, Berkeley, CA-94720, USA.
  • Tallarico JA; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Schirle M; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
  • Toste FD; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Nomura DK; Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, CA-94720, USA.
Chembiochem ; 24(11): e202300116, 2023 06 01.
Article en En | MEDLINE | ID: mdl-37069799

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: SARS-CoV-2 / COVID-19 Límite: Humans Idioma: En Revista: Chembiochem Asunto de la revista: BIOQUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Alemania

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: SARS-CoV-2 / COVID-19 Límite: Humans Idioma: En Revista: Chembiochem Asunto de la revista: BIOQUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Alemania