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SAR study of piperidine derivatives as inhibitors of 1,4-dihydroxy-2-naphthoate isoprenyltransferase (MenA) from Mycobacterium tuberculosis.
Berg, Kaja; Hegde, Pooja; Pujari, Venugopal; Brinkmann, Marzena; Wilkins, David Z; Parish, Tanya; Crick, Dean C; Aldrich, Courtney C.
Afiliación
  • Berg K; Department of Medicinal Chemistry, University of Minnesota, 308 Harvard Street Southeast, Minneapolis, MN, 55455, USA.
  • Hegde P; Department of Medicinal Chemistry, University of Minnesota, 308 Harvard Street Southeast, Minneapolis, MN, 55455, USA.
  • Pujari V; Mycobacteria Research Laboratories, Microbiology, Immunology, and Pathology Department, Colorado State University, Fort Collins, CO, 80523, USA.
  • Brinkmann M; Department of Medicinal Chemistry, University of Minnesota, 308 Harvard Street Southeast, Minneapolis, MN, 55455, USA.
  • Wilkins DZ; Center for Global Infectious Disease Research, Seattle Children's Research Institute, Seattle, WA, 98109, USA.
  • Parish T; Center for Global Infectious Disease Research, Seattle Children's Research Institute, Seattle, WA, 98109, USA.
  • Crick DC; Mycobacteria Research Laboratories, Microbiology, Immunology, and Pathology Department, Colorado State University, Fort Collins, CO, 80523, USA. Electronic address: Dean.Crick@colostate.edu.
  • Aldrich CC; Department of Medicinal Chemistry, University of Minnesota, 308 Harvard Street Southeast, Minneapolis, MN, 55455, USA. Electronic address: aldri015@umn.edu.
Eur J Med Chem ; 249: 115125, 2023 Mar 05.
Article en En | MEDLINE | ID: mdl-36682292

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Tuberculosis / Mycobacterium tuberculosis Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Tuberculosis / Mycobacterium tuberculosis Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Francia