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Lengthening the Guanidine-Aryl Linker of Phenylpyrimidinylguanidines Increases Their Potency as Inhibitors of FOXO3-Induced Gene Transcription.
Kohoutova, Klara; Docekal, Vojtech; Ausserlechner, Michael J; Kaiser, Nora; Tekel, Andrej; Mandal, Raju; Horvath, Matej; Obsilova, Veronika; Vesely, Jan; Hagenbuchner, Judith; Obsil, Tomas.
Afiliación
  • Kohoutova K; Department of Physical and Macromolecular Chemistry, Faculty of Science, Charles University, Albertov 6, Prague 12843, Czech Republic.
  • Docekal V; Institute of Physiology of the Czech Academy of Sciences, Laboratory of Structural Biology of Signaling Proteins, Division BIOCEV, Prumyslova 595, Vestec 25250, Czech Republic.
  • Ausserlechner MJ; Department of Organic Chemistry, Faculty of Science, Charles University, Albertov 6, Prague 12843, Czech Republic.
  • Kaiser N; Department of Pediatrics I, Medical University Innsbruck, Innrain 66, Innsbruck 6020, Austria.
  • Tekel A; Department of Pediatrics I, Medical University Innsbruck, Innrain 66, Innsbruck 6020, Austria.
  • Mandal R; Department of Physical and Macromolecular Chemistry, Faculty of Science, Charles University, Albertov 6, Prague 12843, Czech Republic.
  • Horvath M; Department of Physical and Macromolecular Chemistry, Faculty of Science, Charles University, Albertov 6, Prague 12843, Czech Republic.
  • Obsilova V; Department of Physical and Macromolecular Chemistry, Faculty of Science, Charles University, Albertov 6, Prague 12843, Czech Republic.
  • Vesely J; Institute of Physiology of the Czech Academy of Sciences, Laboratory of Structural Biology of Signaling Proteins, Division BIOCEV, Prumyslova 595, Vestec 25250, Czech Republic.
  • Hagenbuchner J; Department of Organic Chemistry, Faculty of Science, Charles University, Albertov 6, Prague 12843, Czech Republic.
  • Obsil T; Department of Pediatrics II, Medical University Innsbruck, Innrain 66, Innsbruck 6020, Austria.
ACS Omega ; 7(38): 34632-34646, 2022 Sep 27.
Article en En | MEDLINE | ID: mdl-36188303

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Tipo de estudio: Prognostic_studies Idioma: En Revista: ACS Omega Año: 2022 Tipo del documento: Article País de afiliación: República Checa Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Tipo de estudio: Prognostic_studies Idioma: En Revista: ACS Omega Año: 2022 Tipo del documento: Article País de afiliación: República Checa Pais de publicación: Estados Unidos