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Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as PfeEF2.
Laleu, Benoît; Rubiano, Kelly; Yeo, Tomas; Hallyburton, Irene; Anderson, Mark; Crespo-Fernandez, Benigno; Gamo, Francisco-Javier; Antonova-Koch, Yevgeniya; Orjuela-Sanchez, Pamela; Wittlin, Sergio; Jana, Gouranga P; Maity, Bikash C; Chenu, Elodie; Duffy, James; Sjö, Peter; Waterson, David; Winzeler, Elizabeth; Guantai, Eric; Fidock, David A; Hansson, Thomas G.
Afiliación
  • Laleu B; Medicines for Malaria Venture, International Centre Cointrin, Route de Pré-Bois 20, P.O. Box 1826, 1215, Geneva 15, Switzerland.
  • Rubiano K; Department of Microbiology & Immunology, Columbia University Irving Medical Center, New York, NY, 10032, USA.
  • Yeo T; Current address, Department of Molecular Microbiology, Washington University School of Medicine, Saint Louis, MO, 63110, USA.
  • Hallyburton I; Department of Microbiology & Immunology, Columbia University Irving Medical Center, New York, NY, 10032, USA.
  • Anderson M; Drug Discovery Unit, Wellcome Centre for Anti-infective Research, University of Dundee, Dow Street, Dundee, DD1 5EH, UK.
  • Crespo-Fernandez B; Drug Discovery Unit, Wellcome Centre for Anti-infective Research, University of Dundee, Dow Street, Dundee, DD1 5EH, UK.
  • Gamo FJ; Global Health, GlaxoSmithKline R&D, Tres Cantos, 28760, Madrid, Spain.
  • Antonova-Koch Y; Global Health, GlaxoSmithKline R&D, Tres Cantos, 28760, Madrid, Spain.
  • Orjuela-Sanchez P; Department of Pediatrics, School of Medicine, University of California San Diego, La Jolla, CA, 92093, USA.
  • Wittlin S; Current address, Calibr, A Division of Scripps Research, 11119 North Torrey Pines Road, La Jola, CA, 92037, USA.
  • Jana GP; Department of Pediatrics, School of Medicine, University of California San Diego, La Jolla, CA, 92093, USA.
  • Maity BC; Current address, Novartis Institute for Tropical Diseases, 5959 Horton Street, 8th floor, Emeryville, CS, 94608, USA.
  • Chenu E; Swiss Tropical and Public Health Institute, Socinstrasse 57, 4002, Basel, Switzerland.
  • Duffy J; University of Basel, 4002, Basel, Switzerland.
  • Sjö P; TCG Lifesciences Private Limited, Block BN, Plot 7 Salt-lake Electronics Complex, Sector V, Kolkata, 700091, West Bengal, India.
  • Waterson D; TCG Lifesciences Private Limited, Block BN, Plot 7 Salt-lake Electronics Complex, Sector V, Kolkata, 700091, West Bengal, India.
  • Winzeler E; Medicines for Malaria Venture, International Centre Cointrin, Route de Pré-Bois 20, P.O. Box 1826, 1215, Geneva 15, Switzerland.
  • Guantai E; Medicines for Malaria Venture, International Centre Cointrin, Route de Pré-Bois 20, P.O. Box 1826, 1215, Geneva 15, Switzerland.
  • Fidock DA; Medicines for Malaria Venture, International Centre Cointrin, Route de Pré-Bois 20, P.O. Box 1826, 1215, Geneva 15, Switzerland.
  • Hansson TG; Medicines for Malaria Venture, International Centre Cointrin, Route de Pré-Bois 20, P.O. Box 1826, 1215, Geneva 15, Switzerland.
ChemMedChem ; 17(22): e202200393, 2022 11 18.
Article en En | MEDLINE | ID: mdl-36129427

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Malaria Falciparum / Malaria / Antimaláricos Tipo de estudio: Diagnostic_studies / Prognostic_studies Límite: Humans Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2022 Tipo del documento: Article País de afiliación: Suiza Pais de publicación: Alemania

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Malaria Falciparum / Malaria / Antimaláricos Tipo de estudio: Diagnostic_studies / Prognostic_studies Límite: Humans Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2022 Tipo del documento: Article País de afiliación: Suiza Pais de publicación: Alemania