Arenesulfonyl indole: new precursor for diversification of C-3 functionalized indoles.

Kaur, Banni Preet; Kaur, Jasneet; Chimni, Swapandeep Singh

Kaur, Banni Preet; Kaur, Jasneet; Chimni, Swapandeep Singh.

Afiliación

Kaur BP; Department of Chemistry, U.G.C. Centre of Advance Study-II, Guru Nanak Dev University Amritsar Punjab India sschimni@yahoo.com sschimni.chem@gndu.ac.in.
Kaur J; Post-Graduate Department of Chemistry, Khalsa College Amritsar Punjab India jasneet208@gmail.com.
Chimni SS; Department of Chemistry, U.G.C. Centre of Advance Study-II, Guru Nanak Dev University Amritsar Punjab India sschimni@yahoo.com sschimni.chem@gndu.ac.in.

RSC Adv ; 11(4): 2126-2140, 2021 Jan 06.

Article en En | MEDLINE | ID: mdl-35424187

RESUMEN

Arenesulfonyl indoles, bearing a good leaving group, are effective precursors for vinylogous imine intermediates which are generated in situ under basic conditions. This intermediate can readily react with other nucleophilic reagents to obtain C-3 substituted indole derivatives. In the last few years, a plethora of exciting synthetic applications of this substrate have been exploited. The stability of arylsulfonyl-containing substrates, mild reaction conditions, and the large variety of nucleophiles involved in these procedures are the key to their success in organic synthesis.

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Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: RSC Adv Año: 2021 Tipo del documento: Article Pais de publicación: Reino Unido

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