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NLX-112, a highly selective 5-HT1A receptor biased agonist, does not exhibit misuse potential in male rats or macaques.
Depoortère, R; Bergman, J; Beardsley, P M; Desai, R I; Paronis, C A; Walentiny, D M; Varney, M A; Newman-Tancredi, A.
Afiliación
  • Depoortère R; Neurolixis SAS, 2 rue Georges Charpak, 81100, Castres, France. Electronic address: rdepoortere@neurolixis.com.
  • Bergman J; McLean Hospital, Behavioral Biology Program, Belmont, MA, 02478, USA.
  • Beardsley PM; Department of Pharmacology & Toxicology, Virginia Commonwealth University, Richmond, VA, 23298-0613, USA; Center for Biomarker Research and Precision Medicine, Virginia Commonwealth University, Richmond, VA, 23298-0613, USA.
  • Desai RI; McLean Hospital, Behavioral Biology Program, Belmont, MA, 02478, USA.
  • Paronis CA; McLean Hospital, Behavioral Biology Program, Belmont, MA, 02478, USA.
  • Walentiny DM; Department of Pharmacology & Toxicology, Virginia Commonwealth University, Richmond, VA, 23298-0613, USA.
  • Varney MA; Neurolixis SAS, 2 rue Georges Charpak, 81100, Castres, France.
  • Newman-Tancredi A; Neurolixis SAS, 2 rue Georges Charpak, 81100, Castres, France.
Neuropharmacology ; 210: 109025, 2022 06 01.
Article en En | MEDLINE | ID: mdl-35276118

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piperidinas / Piridinas / Agonistas del Receptor de Serotonina 5-HT1 / Macaca Límite: Animals / Humans / Male Idioma: En Revista: Neuropharmacology Año: 2022 Tipo del documento: Article Pais de publicación: Reino Unido

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piperidinas / Piridinas / Agonistas del Receptor de Serotonina 5-HT1 / Macaca Límite: Animals / Humans / Male Idioma: En Revista: Neuropharmacology Año: 2022 Tipo del documento: Article Pais de publicación: Reino Unido