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Rational design of a new near-infrared fluorophore and apply to the detection and imaging study of cysteine and thiophenol.
Yang, Qing-Qing; Ji, Nan; Zhan, Yu; Tian, Qin-Qin; Cai, Ze-Dong; Lu, Xian-Lin; He, Wei.
Afiliación
  • Yang QQ; Department of Chemistry, School of Pharmacy, The Fourth Military Medical University, 169 Changle West Road, Xi'an, 710032, PR China.
  • Ji N; Department of Chemistry, School of Pharmacy, The Fourth Military Medical University, 169 Changle West Road, Xi'an, 710032, PR China.
  • Zhan Y; Department of Chemistry, School of Pharmacy, The Fourth Military Medical University, 169 Changle West Road, Xi'an, 710032, PR China.
  • Tian QQ; Department of Chemistry, School of Pharmacy, The Fourth Military Medical University, 169 Changle West Road, Xi'an, 710032, PR China.
  • Cai ZD; Department of Pharmaceutics, School of Pharmacy, The Fourth Military Medical University, Xi'an, 710032, PR China.
  • Lu XL; Department of Chemistry, School of Pharmacy, The Fourth Military Medical University, 169 Changle West Road, Xi'an, 710032, PR China.
  • He W; Department of Chemistry, School of Pharmacy, The Fourth Military Medical University, 169 Changle West Road, Xi'an, 710032, PR China. Electronic address: weihechem@fmmu.edu.cn.
Anal Chim Acta ; 1186: 339116, 2021 Nov 22.
Article en En | MEDLINE | ID: mdl-34756262
The development of a near-infrared fluorophore with excellent fluorescence performance, a large Stokes shift, and good biocompatibility has become a focus in the field of fluorescence imaging in recent years. Based on quantum chemistry calculations and reasonable molecular design strategies, a new NIR fluorophore was developed and characterized by simple synthesis, easy structural modification, and a large Stokes shift (105 nm). Furthermore, two new "activatable" fluorescent probes QN-Cys and QN-DNP were synthesized using a simple structural modification. The probe QN-Cys can recognize Cys with high sensitivity (LOD = 128 nM) and high selectivity, and its fluorescence intensity has a good linear relationship with the Cys concentration in the range of 5-35 µM. Furthermore, probe QN-Cys can effectively distinguish Cys from Hcy and GSH, and was successfully applied to the detection and imaging of Cys in human serum, cells, and zebrafish. The probe QN-DNP showed a good specific and sensitive (LOD = 78 nM) fluorescence response to thiophenol, and its fluorescence intensity has a good linear relationship with the thiophenol concentration in the range of 5-30 µM. Furthermore, it was successfully applied to detect thiophenol in real water samples with good recoveries (97-102%), and image thiophenol in living cells, zebrafish and mice. Notebly, the QN-DNP probe could be applied to visualize the distribution of thiophenol in the mice.
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Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Cisteína / Colorantes Fluorescentes Tipo de estudio: Diagnostic_studies Límite: Animals / Humans Idioma: En Revista: Anal Chim Acta Año: 2021 Tipo del documento: Article Pais de publicación: Países Bajos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Cisteína / Colorantes Fluorescentes Tipo de estudio: Diagnostic_studies Límite: Animals / Humans Idioma: En Revista: Anal Chim Acta Año: 2021 Tipo del documento: Article Pais de publicación: Países Bajos