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Discovery of the Selective Protein Kinase C-θ Kinase Inhibitor, CC-90005.
Papa, Patrick; Whitefield, Brandon; Mortensen, Deborah S; Cashion, Dan; Huang, Dehua; Torres, Eduardo; Parnes, Jason; Sapienza, John; Hansen, Joshua; Correa, Matthew; Delgado, Mercedes; Harris, Roy; Hegde, Sayee; Norris, Stephen; Bahmanyar, Sogole; Plantevin-Krenitsky, Veronique; Liu, Zheng; Leftheris, Katerina; Kulkarni, Ashutosh; Bennett, Brydon; Hur, Eun Mi; Ringheim, Garth; Khambatta, Godrej; Chan, Henry; Muir, Jeffrey; Blease, Kate; Burnett, Kelven; LeBrun, Laurie; Morrison, Lisa; Celeridad, Maria; Khattri, Roli; Cathers, Brian E.
Afiliación
  • Papa P; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Whitefield B; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Mortensen DS; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Cashion D; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Huang D; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Torres E; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Parnes J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Sapienza J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Hansen J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Correa M; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Delgado M; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Harris R; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Hegde S; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Norris S; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Bahmanyar S; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Plantevin-Krenitsky V; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Liu Z; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Leftheris K; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Kulkarni A; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Bennett B; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Hur EM; Bristol Myers Squibb, 86 Morris Avenue, Summit, New Jersey 07901, United States.
  • Ringheim G; Bristol Myers Squibb, 86 Morris Avenue, Summit, New Jersey 07901, United States.
  • Khambatta G; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Chan H; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Muir J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Blease K; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Burnett K; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • LeBrun L; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Morrison L; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Celeridad M; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Khattri R; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Cathers BE; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
J Med Chem ; 64(16): 11886-11903, 2021 08 26.
Article en En | MEDLINE | ID: mdl-34355886

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pirimidinas / Ciclohexanoles / Inhibidores de Proteínas Quinasas / Proteína Quinasa C-theta / Enfermedad Injerto contra Huésped / Factores Inmunológicos Tipo de estudio: Prognostic_studies Límite: Animals / Humans / Male Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pirimidinas / Ciclohexanoles / Inhibidores de Proteínas Quinasas / Proteína Quinasa C-theta / Enfermedad Injerto contra Huésped / Factores Inmunológicos Tipo de estudio: Prognostic_studies Límite: Animals / Humans / Male Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos