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Submicron particle docetaxel intratumoral injection in combination with anti-mCTLA-4 into 4T1-Luc orthotopic implants reduces primary tumor and metastatic pulmonary lesions.
Maulhardt, Holly; Marin, Alyson; Hesseltine, Holly; diZerega, Gere.
Afiliación
  • Maulhardt H; US Biotest, Inc., 231 Bonetti Drive, Suite 240, San Luis Obispo, CA, USA.
  • Marin A; US Biotest, Inc., 231 Bonetti Drive, Suite 240, San Luis Obispo, CA, USA.
  • Hesseltine H; US Biotest, Inc., 231 Bonetti Drive, Suite 240, San Luis Obispo, CA, USA.
  • diZerega G; US Biotest, Inc., 231 Bonetti Drive, Suite 240, San Luis Obispo, CA, USA. gere.dizerega@usbiotest.com.
Med Oncol ; 38(9): 106, 2021 Jul 31.
Article en En | MEDLINE | ID: mdl-34331595
We describe here characterization of the response of local and metastatic disease and immunomodulation following intratumoral (IT) injection of submicron particle docetaxel (SPD) administered alone or in combination with systemic antibody anti-mCTLA-4 (anti-mCTLA-4) in the metastatic 4T1-Luc2-1A4 (4T1) murine breast cancer model. In-life assessments of treatment tolerance, tumor volume (TV), and metastasis were performed (n = 10 animals/group). At study end, immune cell populations in tumor-site tissues and peripheral blood were analyzed using flow cytometry. Signs of distress typical of this aggressive tumor model occurred across all animals except for the combination treated which were asymptomatic and gained weight. TV at study end was significantly reduced in the combination group versus untreated [43% reduced (p < 0.05)] and vehicle controls [54% reduced (p < 0.0001)]. No evidence of thoracic metastasis was found in 40% of combination group animals and thoracic bioluminescence imaging (BLI) was reduced vs. untreated controls (p < 0.01). Significant elevations (p < 0.05) in CD4 + T, CD4 + helper T, Treg, and NKT cells were found in tumor and blood in SPD or combination treatment compared to controls or anti-mCTLA-4. Combination treatment increased tumor-associated CD8 + T cells (p < 0.01), peripheral B cells (p < 0.01), and tumor associated and circulating dendritic cells (DC) (p < 0.05). Tumor-associated NK cells were significantly increased in SPD ± anti-mCTLA-4 treatments (p < 0.01). Myeloid-derived suppressor cells (MDSC) were reduced in bloods in SPD ± anti-mCTLA-4 groups (p < 0.05). These data demonstrate that both SPD and anti-mCTLA-4 produce local anti-tumor effects as well as reductions in metastasis which are significantly enhanced when administered in combination.
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Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Neoplasias Mamarias Animales / Linfocitos Infiltrantes de Tumor / Antígeno CTLA-4 / Docetaxel / Inhibidores de Puntos de Control Inmunológico / Neoplasias Pulmonares / Anticuerpos Monoclonales Límite: Animals Idioma: En Revista: Med Oncol Asunto de la revista: NEOPLASIAS Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Neoplasias Mamarias Animales / Linfocitos Infiltrantes de Tumor / Antígeno CTLA-4 / Docetaxel / Inhibidores de Puntos de Control Inmunológico / Neoplasias Pulmonares / Anticuerpos Monoclonales Límite: Animals Idioma: En Revista: Med Oncol Asunto de la revista: NEOPLASIAS Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos