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Pharmacodynamic and pharmacokinetic profiles of a neurotensin receptor type 2 (NTS2) analgesic macrocyclic analog.
Chartier, Magali; Desgagné, Michael; Sousbie, Marc; Rumsby, Charles; Chevillard, Lucie; Théroux, Léa; Haroune, Lounès; Côté, Jérôme; Longpré, Jean-Michel; Boudreault, Pierre-Luc; Marsault, Éric; Sarret, Philippe.
Afiliación
  • Chartier M; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Magali.Chartier@USherbrooke.ca.
  • Desgagné M; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Michael.Desgagne@USherbrooke.ca.
  • Sousbie M; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Marc.Sousbie@USherbrooke.ca.
  • Rumsby C; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Charles.Rumsby@USherbrooke.ca.
  • Chevillard L; Inserm, UMR-S 1144, Université de Paris, Paris, France. Electronic address: luciechevillard@gmail.com.
  • Théroux L; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Lea.Theroux@USherbrooke.ca.
  • Haroune L; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Lounes.Haroune@USherbrooke.ca.
  • Côté J; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Jerome.Cote@USherbrooke.ca.
  • Longpré JM; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Jean-Michel.Longpre@USherbrooke.ca.
  • Boudreault PL; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Pierre-Luc.Boudreault@USherbrooke.ca.
  • Marsault É; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: Philippe.Sarret@USherbrooke.ca.
  • Sarret P; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC, Canada. Electronic address: philippe.sarret@usherbrooke.ca.
Biomed Pharmacother ; 141: 111861, 2021 Sep.
Article en En | MEDLINE | ID: mdl-34229249

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Receptores de Neurotensina / Analgésicos no Narcóticos / Compuestos Macrocíclicos Tipo de estudio: Etiology_studies Límite: Animals Idioma: En Revista: Biomed Pharmacother Año: 2021 Tipo del documento: Article Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Receptores de Neurotensina / Analgésicos no Narcóticos / Compuestos Macrocíclicos Tipo de estudio: Etiology_studies Límite: Animals Idioma: En Revista: Biomed Pharmacother Año: 2021 Tipo del documento: Article Pais de publicación: Francia