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Synthesis of HDAC Inhibitor Libraries via Microscale Workflow.
Dykstra, Kevin D; Streckfuss, Eric; Liu, Min; Liu, Jian; Yu, Younong; Wang, Ming; Kozlowski, Joseph A; Myers, Robert W; Buevich, Alexei V; Maletic, Milana M; Vachal, Petr; Krska, Shane W.
Afiliación
  • Dykstra KD; Chemical Capabilities for Accelerating Therapeutics, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Streckfuss E; Discovery Chemistry, Merck & Co., Inc., West Point, Pennsylvania 19486, United States.
  • Liu M; Chemical Capabilities for Accelerating Therapeutics, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Liu J; Screening, Targets and Compound Profiling, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Yu Y; Chemical Capabilities for Accelerating Therapeutics, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Wang M; Chemical Capabilities for Accelerating Therapeutics, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Kozlowski JA; Discovery Chemistry, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Myers RW; Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Buevich AV; NMR Structure Elucidation, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Maletic MM; Chemical Capabilities for Accelerating Therapeutics, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Vachal P; Screening, Targets and Compound Profiling, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
  • Krska SW; Chemical Capabilities for Accelerating Therapeutics, Merck & Co., Inc., Kenilworth, New Jersey 07033, United States.
ACS Med Chem Lett ; 12(3): 337-342, 2021 Mar 11.
Article en En | MEDLINE | ID: mdl-33738059

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos