Your browser doesn't support javascript.
loading
Optical porosimetry by gas in scattering media absorption spectroscopy (GASMAS) applied to roller compaction ribbons.
Johansson, Jonas; Sparén, Anders; Wikström, Håkan; Tajarobi, Pirjo; Koch, Roland; Lundin, Patrik; Långberg, Anders; Sebesta, Mikael; Lewander Xu, Märta.
Afiliación
  • Johansson J; Innovation Strategies & External Liaison, Pharmaceutical Technology & Development, Operations, AstraZeneca, Gothenburg, Sweden. Electronic address: jonas.johansson@astrazeneca.com.
  • Sparén A; Oral Product Development, Pharmaceutical Technology & Development, Operations, AstraZeneca, Gothenburg, Sweden.
  • Wikström H; Oral Product Development, Pharmaceutical Technology & Development, Operations, AstraZeneca, Gothenburg, Sweden.
  • Tajarobi P; Early Product Development & Manufacturing, Pharmaceutical Sciences, BioPharmaceuticals R&D, AstraZeneca, Gothenburg, Sweden.
  • Koch R; Gasporox AB, Maskinvägen 1, S-22730 Lund, Sweden.
  • Lundin P; Gasporox AB, Maskinvägen 1, S-22730 Lund, Sweden.
  • Långberg A; Gasporox AB, Maskinvägen 1, S-22730 Lund, Sweden.
  • Sebesta M; Gasporox AB, Maskinvägen 1, S-22730 Lund, Sweden.
  • Lewander Xu M; Gasporox AB, Maskinvägen 1, S-22730 Lund, Sweden.
Int J Pharm ; 592: 120056, 2021 Jan 05.
Article en En | MEDLINE | ID: mdl-33161035
Currently, there is a need for new technology for in-line or fast at-line assessment of solid material porosity. One specific gap is a fast technology to be used in connection to roller compaction (RC) manufacturing, where the porosity of the RC ribbons is critical to the manufacturing of tablets of the right tensile strength and disintegration properties. In this paper, the development of an at-line technology for fast, non-destructive assessment of porosity of RC ribbons is reported. The technology is based on a diode laser spectroscopic technique called Gas in scattering media absorption spectroscopy (GASMAS). GASMAS measures the sample voids by laser light, giving the distance through air. The total distance the light travels is measured using time-of-flight spectroscopy (TOFS). The ratio of these measures gives an "optical porosity", which through theory relates to the porosity of the sample. We present a description of the technology, evaluations of measurement robustness and results from an experimental design where roller compactor, roll force, roll gap and formulation were varied. It is concluded that the data from two different pharmaceutical formulations is supported by the same calibration curve, which indicates that optical porosimetry is a general technique for pharmaceutical materials that does not require frequent calibrations.
Asunto(s)
Palabras clave

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Tecnología Farmacéutica / Gases Idioma: En Revista: Int J Pharm Año: 2021 Tipo del documento: Article Pais de publicación: Países Bajos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Tecnología Farmacéutica / Gases Idioma: En Revista: Int J Pharm Año: 2021 Tipo del documento: Article Pais de publicación: Países Bajos