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Determination of the inhibition profiles of pyrazolyl-thiazole derivatives against aldose reductase and α-glycosidase and molecular docking studies.
Demir, Yeliz; Taslimi, Parham; Koçyigit, Ümit M; Akkus, Musa; Özaslan, Muhammet Serhat; Duran, Hatice Esra; Budak, Yakup; Tüzün, Burak; Gürdere, Meliha B; Ceylan, Mustafa; Taysi, Seyithan; Gülçin, Ilhami; Beydemir, Sükrü.
Afiliación
  • Demir Y; Department of Pharmacy Services, Nihat Delibalta Göle Vocational High School, Ardahan University, Ardahan, Turkey.
  • Taslimi P; Department of Biotechnology, Faculty of Science, Bartin University, Bartin, Turkey.
  • Koçyigit ÜM; Department of Basic Pharmaceutical Sciences, Division of Biochemistry, Faculty of Pharmacy, Cumhuriyet University, Sivas, Turkey.
  • Akkus M; Department of Chemistry, Faculty of Science, Atatürk University, Erzurum, Turkey.
  • Özaslan MS; Department of Pharmacy Services, Nihat Delibalta Göle Vocational High School, Ardahan University, Ardahan, Turkey.
  • Duran HE; Department of Biochemistry, Medical School, Kafkas University, Kars, Turkey.
  • Budak Y; Department of Chemistry, Faculty of Arts and Sciences, Gaziosmanpasa University, Tokat, Turkey.
  • Tüzün B; Department of Chemistry, Faculty of Science, Cumhuriyet University, Sivas, Turkey.
  • Gürdere MB; Department of Chemistry, Faculty of Arts and Sciences, Gaziosmanpasa University, Tokat, Turkey.
  • Ceylan M; Department of Chemistry, Faculty of Arts and Sciences, Gaziosmanpasa University, Tokat, Turkey.
  • Taysi S; Department of Biochemistry and Clinical Biochemistry, Medical School, Gaziantep University, Gaziantep, Turkey.
  • Gülçin I; Department of Chemistry, Faculty of Science, Atatürk University, Erzurum, Turkey.
  • Beydemir S; Department of Biochemistry, Faculty of Pharmacy, Anadolu University, Eskisehir, Turkey.
Arch Pharm (Weinheim) ; 353(12): e2000118, 2020 Dec.
Article en En | MEDLINE | ID: mdl-32761859

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pirazoles / Tiazoles / Aldehído Reductasa / Inhibidores Enzimáticos / Simulación del Acoplamiento Molecular / Glicósido Hidrolasas / Hipoglucemiantes Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Revista: Arch Pharm (Weinheim) Año: 2020 Tipo del documento: Article País de afiliación: Turquía Pais de publicación: Alemania

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pirazoles / Tiazoles / Aldehído Reductasa / Inhibidores Enzimáticos / Simulación del Acoplamiento Molecular / Glicósido Hidrolasas / Hipoglucemiantes Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Revista: Arch Pharm (Weinheim) Año: 2020 Tipo del documento: Article País de afiliación: Turquía Pais de publicación: Alemania