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Optimizing the aryl-triazole of cjoc42 for enhanced gankyrin binding and anti-cancer activity.
Kanabar, Dipti; Farrales, Pamela; Kabir, Abbas; Juang, Daniel; Gnanmony, Manu; Almasri, Joseph; Torrents, Nicolas; Shukla, Snehal; Gupta, Vivek; Dukhande, Vikas V; D'Souza, Amber; Muth, Aaron.
Afiliación
  • Kanabar D; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, NY 11439, USA.
  • Farrales P; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, NY 11439, USA.
  • Kabir A; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, NY 11439, USA.
  • Juang D; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, NY 11439, USA.
  • Gnanmony M; Department of Pediatrics, Hematology and Oncology, University of Illinois College of Medicine, Chicago, IL 60612, USA.
  • Almasri J; Department of Chemistry, College of Liberal Arts and Sciences, St. John's University, Queens, NY 11439, USA.
  • Torrents N; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, NY 11439, USA.
  • Shukla S; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, NY 11439, USA.
  • Gupta V; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, NY 11439, USA.
  • Dukhande VV; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, NY 11439, USA.
  • D'Souza A; Department of Pediatrics, Hematology and Oncology, University of Illinois College of Medicine, Chicago, IL 60612, USA.
  • Muth A; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, St. John's University, Queens, NY 11439, USA.
Bioorg Med Chem Lett ; 30(17): 127372, 2020 09 01.
Article en En | MEDLINE | ID: mdl-32738965

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Triazoles / Bencenosulfonatos / Proteínas Proto-Oncogénicas / Complejo de la Endopetidasa Proteasomal / Antineoplásicos Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Reino Unido

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Triazoles / Bencenosulfonatos / Proteínas Proto-Oncogénicas / Complejo de la Endopetidasa Proteasomal / Antineoplásicos Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Reino Unido