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Novel bacterial topoisomerase inhibitors derived from isomannide.
Okumu, Antony; Lu, Yanran; Dellos-Nolan, Sheri; Papa, Jonathan L; Koci, Bryan; Cockroft, Nicholas T; Gallucci, Judith; Wozniak, Daniel J; Yalowich, Jack C; Mitton-Fry, Mark J.
Afiliación
  • Okumu A; Division of Medicinal Chemistry and Pharmacognosy. The Ohio State University, Columbus, OH, 43210, USA.
  • Lu Y; Division of Medicinal Chemistry and Pharmacognosy. The Ohio State University, Columbus, OH, 43210, USA.
  • Dellos-Nolan S; Microbial Infection and Immunity. The Ohio State University, Columbus, OH, 43210, USA.
  • Papa JL; Division of Pharmaceutics and Pharmacology. The Ohio State University, Columbus, OH, 43210, USA.
  • Koci B; Eurofins Panlabs. St. Charles, MO, 63304, USA.
  • Cockroft NT; Division of Medicinal Chemistry and Pharmacognosy. The Ohio State University, Columbus, OH, 43210, USA.
  • Gallucci J; Department of Chemistry and Biochemistry. The Ohio State University, Columbus, OH, 43210, USA.
  • Wozniak DJ; Microbial Infection and Immunity. The Ohio State University, Columbus, OH, 43210, USA; Department of Microbiology. The Ohio State University, Columbus, OH, 43210, USA.
  • Yalowich JC; Division of Pharmaceutics and Pharmacology. The Ohio State University, Columbus, OH, 43210, USA.
  • Mitton-Fry MJ; Division of Medicinal Chemistry and Pharmacognosy. The Ohio State University, Columbus, OH, 43210, USA. Electronic address: mitton-fry.1@osu.edu.
Eur J Med Chem ; 199: 112324, 2020 Aug 01.
Article en En | MEDLINE | ID: mdl-32402932

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Compuestos Bicíclicos Heterocíclicos con Puentes / Inhibidores de Topoisomerasa / Bacterias Grampositivas / Antibacterianos Idioma: En Revista: Eur J Med Chem Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Compuestos Bicíclicos Heterocíclicos con Puentes / Inhibidores de Topoisomerasa / Bacterias Grampositivas / Antibacterianos Idioma: En Revista: Eur J Med Chem Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Francia