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Discovery of 5-naphthylidene-2,4-thiazolidinedione derivatives as selective HDAC8 inhibitors and evaluation of their cytotoxic effects in leukemic cell lines.
Tilekar, Kalpana; Upadhyay, Neha; Jänsch, Niklas; Schweipert, Markus; Mrowka, Piotr; Meyer-Almes, F J; Ramaa, C S.
Afiliación
  • Tilekar K; Department of Pharmaceutical Chemistry, Bharati Vidyapeeth's College of Pharmacy, Navi Mumbai, Maharashtra, India.
  • Upadhyay N; Department of Pharmaceutical Chemistry, Bharati Vidyapeeth's College of Pharmacy, Navi Mumbai, Maharashtra, India.
  • Jänsch N; Department of Chemical Engineering and Biotechnology, University of Applied Sciences, Darmstadt, Germany.
  • Schweipert M; Department of Chemical Engineering and Biotechnology, University of Applied Sciences, Darmstadt, Germany.
  • Mrowka P; Department of Biophysics and Human Physiology, Medical University of Warsaw, Chalubinskiego, Warsaw, Poland.
  • Meyer-Almes FJ; Department of Chemical Engineering and Biotechnology, University of Applied Sciences, Darmstadt, Germany. Electronic address: franz-josef.meyer-almes@h-da.de.
  • Ramaa CS; Department of Pharmaceutical Chemistry, Bharati Vidyapeeth's College of Pharmacy, Navi Mumbai, Maharashtra, India. Electronic address: sinharamaa@yahoo.in.
Bioorg Chem ; 95: 103522, 2020 01.
Article en En | MEDLINE | ID: mdl-31901516

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Proteínas Represoras / Tiazolidinedionas / Inhibidores Enzimáticos / Descubrimiento de Drogas / Antineoplásicos Límite: Humans Idioma: En Revista: Bioorg Chem Año: 2020 Tipo del documento: Article País de afiliación: India Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Proteínas Represoras / Tiazolidinedionas / Inhibidores Enzimáticos / Descubrimiento de Drogas / Antineoplásicos Límite: Humans Idioma: En Revista: Bioorg Chem Año: 2020 Tipo del documento: Article País de afiliación: India Pais de publicación: Estados Unidos