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Large-scale High-throughput Screening Revealed 5'-(carbonylamino)-2,3'- bithiophene-4'-carboxylate as Novel Template for Antibacterial Agents.
Ivanenkov, Yan A; Yamidanov, Renat S; Osterman, Ilya A; Sergiev, Petr V; Aladinskiy, Vladimir A; Aladinskaya, Anastasia V; Terentiev, Victor A; Veselov, Mark S; Ayginin, Andrey A; Skvortsov, Dmitry A; Komarova, Katerina S; Zagribelnyy, Bogdan A; Baimiev, Alexey Kh; Shvetc, Kseniya Yu; Baimiev, Andrey Kh; Sofronova, Alina A; Machulkin, Alexey E; Petrov, Rostislav A; Zainullina, Liana F; Maximova, Marina A; Zileeva, Zulfiya R; Vakhitova, Yulia V; Bezrukov, Dmitry S; Puchinina, Maria M; Dontsova, Olga A.
Afiliación
  • Ivanenkov YA; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Yamidanov RS; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Osterman IA; Lomonosov Moscow State University, Chemistry Dept, Leninskie gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.
  • Sergiev PV; Skolkovo Institute of Science and Technology, Skolkovo, Russian Federation.
  • Aladinskiy VA; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation.
  • Aladinskaya AV; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation.
  • Terentiev VA; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Veselov MS; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Ayginin AA; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Skvortsov DA; Lomonosov Moscow State University, Department of Chemistry and A.N. Belozersky Institute of Physico-Chemical Biology, Moscow, Russian Federation.
  • Komarova KS; Lomonosov Moscow State University, Department of Chemistry and A.N. Belozersky Institute of Physico-Chemical Biology, Moscow, Russian Federation.
  • Zagribelnyy BA; Lomonosov Moscow State University, Chemistry Dept, Leninskie gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.
  • Baimiev AK; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Shvetc KY; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Baimiev AK; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Sofronova AA; Lomonosov Moscow State University, Faculty of Bioengineering and Bioinformatics, Moscow, Russian Federation.
  • Machulkin AE; Lomonosov Moscow State University, Chemistry Dept, Leninskie gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.
  • Petrov RA; Lomonosov Moscow State University, Chemistry Dept, Leninskie gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.
  • Zainullina LF; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Maximova MA; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Zileeva ZR; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Vakhitova YV; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Bezrukov DS; Lomonosov Moscow State University, Chemistry Dept, Leninskie gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.
  • Puchinina MM; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation.
  • Dontsova OA; Lomonosov Moscow State University, Chemistry Dept, Leninskie gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.
Curr Drug Discov Technol ; 17(5): 716-724, 2020.
Article en En | MEDLINE | ID: mdl-31161993

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Tiofenos / Descubrimiento de Drogas / Ensayos Analíticos de Alto Rendimiento / Antibacterianos Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: Curr Drug Discov Technol Asunto de la revista: FARMACOLOGIA Año: 2020 Tipo del documento: Article Pais de publicación: Emiratos Árabes Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Tiofenos / Descubrimiento de Drogas / Ensayos Analíticos de Alto Rendimiento / Antibacterianos Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: Curr Drug Discov Technol Asunto de la revista: FARMACOLOGIA Año: 2020 Tipo del documento: Article Pais de publicación: Emiratos Árabes Unidos