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A 3-(4-nitronaphthen-1-yl) amino-benzoate analog as a bifunctional AKR1C3 inhibitor and AR antagonist: Head to head comparison with other advanced AKR1C3 targeted therapeutics.
Wangtrakuldee, Phumvadee; Adeniji, Adegoke O; Zang, Tianzhu; Duan, Ling; Khatri, Buddha; Twenter, Barry M; Estrada, Michelle A; Higgins, Tyler F; Winkler, Jeffrey D; Penning, Trevor M.
Afiliación
  • Wangtrakuldee P; Department of Systems Pharmacology and Translational Therapeutics and the Center for Excellence in Environmental Toxicology, Perelman School of Medicine, University of Pennsylvania, 1315 BRBII/III, 421 Curie Boulevard, Philadelphia, PA 19104-6160, USA.
  • Adeniji AO; Department of Systems Pharmacology and Translational Therapeutics and the Center for Excellence in Environmental Toxicology, Perelman School of Medicine, University of Pennsylvania, 1315 BRBII/III, 421 Curie Boulevard, Philadelphia, PA 19104-6160, USA.
  • Zang T; Department of Systems Pharmacology and Translational Therapeutics and the Center for Excellence in Environmental Toxicology, Perelman School of Medicine, University of Pennsylvania, 1315 BRBII/III, 421 Curie Boulevard, Philadelphia, PA 19104-6160, USA.
  • Duan L; Department of Systems Pharmacology and Translational Therapeutics and the Center for Excellence in Environmental Toxicology, Perelman School of Medicine, University of Pennsylvania, 1315 BRBII/III, 421 Curie Boulevard, Philadelphia, PA 19104-6160, USA.
  • Khatri B; Department of Chemistry, University of Pennsylvania, 231 S. 34thStreet, Philadelphia, PA 19104-6323, USA.
  • Twenter BM; Department of Chemistry, University of Pennsylvania, 231 S. 34thStreet, Philadelphia, PA 19104-6323, USA.
  • Estrada MA; Department of Chemistry, University of Pennsylvania, 231 S. 34thStreet, Philadelphia, PA 19104-6323, USA.
  • Higgins TF; Department of Chemistry, University of Pennsylvania, 231 S. 34thStreet, Philadelphia, PA 19104-6323, USA.
  • Winkler JD; Department of Chemistry, University of Pennsylvania, 231 S. 34thStreet, Philadelphia, PA 19104-6323, USA.
  • Penning TM; Department of Systems Pharmacology and Translational Therapeutics and the Center for Excellence in Environmental Toxicology, Perelman School of Medicine, University of Pennsylvania, 1315 BRBII/III, 421 Curie Boulevard, Philadelphia, PA 19104-6160, USA. Electronic address: penning@upenn.edu.
J Steroid Biochem Mol Biol ; 192: 105283, 2019 09.
Article en En | MEDLINE | ID: mdl-30641225
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Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Benzoatos / Receptores Androgénicos / Inhibidores Enzimáticos / Antagonistas de Receptores Androgénicos / Neoplasias de la Próstata Resistentes a la Castración / Miembro C3 de la Familia 1 de las Aldo-Ceto Reductasas / Naftalenos Límite: Humans / Male Idioma: En Revista: J Steroid Biochem Mol Biol Asunto de la revista: BIOLOGIA MOLECULAR / BIOQUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Reino Unido
Texto completo
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Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Benzoatos / Receptores Androgénicos / Inhibidores Enzimáticos / Antagonistas de Receptores Androgénicos / Neoplasias de la Próstata Resistentes a la Castración / Miembro C3 de la Familia 1 de las Aldo-Ceto Reductasas / Naftalenos Límite: Humans / Male Idioma: En Revista: J Steroid Biochem Mol Biol Asunto de la revista: BIOLOGIA MOLECULAR / BIOQUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Reino Unido