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Design, synthesis and antibacterial evaluation of 2,4-disubstituted-6-thiophenyl-pyrimidines.
Fang, Zhiyuan; Zheng, Sichao; Chan, Kin-Fai; Yuan, Wenchang; Guo, Qi; Wu, Wenyu; Lui, Hoi-Kui; Lu, Yujing; Leung, Yun-Chung; Chan, Tak-Hang; Wong, Kwok-Yin; Sun, Ning.
Afiliación
  • Fang Z; The Fifth Affiliated Hospital of Guangzhou Medical University, Guangzhou, 510700, PR China.
  • Zheng S; The Fifth Affiliated Hospital of Guangzhou Medical University, Guangzhou, 510700, PR China.
  • Chan KF; State Key Laboratory of Chemical Biology and Drug Discovery, Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong, China. Electronic address: kf.chan@polyu.edu.hk.
  • Yuan W; The Fifth Affiliated Hospital of Guangzhou Medical University, Guangzhou, 510700, PR China.
  • Guo Q; State Key Laboratory of Ophthalmology, Zhongshan Ophthalmic Center, Sun Yat-sen University, 54 South Xianlie Road, Guangzhou, 510060, PR China.
  • Wu W; State Key Laboratory of Ophthalmology, Zhongshan Ophthalmic Center, Sun Yat-sen University, 54 South Xianlie Road, Guangzhou, 510060, PR China.
  • Lui HK; State Key Laboratory of Chemical Biology and Drug Discovery, Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong, China.
  • Lu Y; Institute of Natural Medicine and Green Chemistry, School of Chemical Engineering and Light Industry, Guangdong University of Technology, Guangzhou, 510006, PR China.
  • Leung YC; State Key Laboratory of Chemical Biology and Drug Discovery, Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong, China.
  • Chan TH; State Key Laboratory of Chemical Biology and Drug Discovery, Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong, China; Department of Chemistry, McGill University, Montreal, Quebec, H3A 2K6, Canada.
  • Wong KY; State Key Laboratory of Chemical Biology and Drug Discovery, Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong, China. Electronic address: kwok-yin.wong@polyu.edu.hk.
  • Sun N; The Fifth Affiliated Hospital of Guangzhou Medical University, Guangzhou, 510700, PR China; State Key Laboratory of Chemical Biology and Drug Discovery, Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong, China. Electronic addres
Eur J Med Chem ; 161: 141-153, 2019 Jan 01.
Article en En | MEDLINE | ID: mdl-30347327

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pirimidinas / Tiofenos / Diseño de Fármacos / Staphylococcus aureus Resistente a Meticilina / Enterococos Resistentes a la Vancomicina / Antibacterianos Idioma: En Revista: Eur J Med Chem Año: 2019 Tipo del documento: Article Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pirimidinas / Tiofenos / Diseño de Fármacos / Staphylococcus aureus Resistente a Meticilina / Enterococos Resistentes a la Vancomicina / Antibacterianos Idioma: En Revista: Eur J Med Chem Año: 2019 Tipo del documento: Article Pais de publicación: Francia