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Cp*Co(iii)-Catalyzed oxidative [5+2] annulation: regioselective synthesis of 2-aminobenzoxepines via C-H/O-H functionalization of 2-vinylphenols with ynamides.
Han, Xiang-Lei; Liu, Xu-Ge; Lin, E; Chen, Yunyun; Chen, Zhuangzhong; Wang, Honggen; Li, Qingjiang.
Afiliación
  • Han XL; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou, 510006, China. liqingj3@mail.sysu.edu.cn.
Chem Commun (Camb) ; 54(82): 11562-11565, 2018 Oct 11.
Article en En | MEDLINE | ID: mdl-30225492
A Cp*Co(iii)-catalyzed [5+2] C-H annulation reaction of 2-vinylphenols with ynamides was developed. The reaction led to the efficient synthesis of valuable 2-aminobenzoxepines in high regioselectivity. Mild reaction conditions, good functional group tolerance, and moderate to good yields were observed. The synthetic utility was demonstrated by a gram-scale synthesis and further transformations of the products. Preliminary mechanistic studies were conducted, and a possible catalytic cycle was proposed.

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: Chem Commun (Camb) Asunto de la revista: QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: China Pais de publicación: Reino Unido

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: Chem Commun (Camb) Asunto de la revista: QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: China Pais de publicación: Reino Unido