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Entry from the Lipid Bilayer: A Possible Pathway for Inhibition of a Peptide G Protein-Coupled Receptor by a Lipophilic Small Molecule.
Bokoch, Michael P; Jo, Hyunil; Valcourt, James R; Srinivasan, Yoga; Pan, Albert C; Capponi, Sara; Grabe, Michael; Dror, Ron O; Shaw, David E; DeGrado, William F; Coughlin, Shaun R.
Afiliación
  • Bokoch MP; Cardiovascular Research Institute , University of California , San Francisco , California 94158 , United States.
  • Jo H; Department of Anesthesia and Perioperative Care , University of California , San Francisco , California 94143 , United States.
  • Valcourt JR; Department of Pharmaceutical Chemistry , University of California , San Francisco , California 94143 , United States.
  • Srinivasan Y; D. E. Shaw Research , New York , New York 10036 , United States.
  • Pan AC; Cardiovascular Research Institute , University of California , San Francisco , California 94158 , United States.
  • Capponi S; D. E. Shaw Research , New York , New York 10036 , United States.
  • Grabe M; Cardiovascular Research Institute , University of California , San Francisco , California 94158 , United States.
  • Dror RO; Cardiovascular Research Institute , University of California , San Francisco , California 94158 , United States.
  • Shaw DE; D. E. Shaw Research , New York , New York 10036 , United States.
  • DeGrado WF; D. E. Shaw Research , New York , New York 10036 , United States.
  • Coughlin SR; Department of Biochemistry and Molecular Biophysics , Columbia University , New York , New York 10032 , United States.
Biochemistry ; 57(39): 5748-5758, 2018 10 02.
Article en En | MEDLINE | ID: mdl-30102523

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piridinas / Receptor PAR-1 / Lactonas / Membrana Dobles de Lípidos Límite: Animals / Humans Idioma: En Revista: Biochemistry Año: 2018 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piridinas / Receptor PAR-1 / Lactonas / Membrana Dobles de Lípidos Límite: Animals / Humans Idioma: En Revista: Biochemistry Año: 2018 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos