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Mathematical and Structural Characterization of Strong Nonadditive Structure-Activity Relationship Caused by Protein Conformational Changes.
Gomez, Laurent; Xu, Rui; Sinko, William; Selfridge, Brandon; Vernier, William; Ly, Kiev; Truong, Richard; Metz, Markus; Marrone, Tami; Sebring, Kristen; Yan, Yingzhou; Appleton, Brent; Aertgeerts, Kathleen; Massari, Mark Eben; Breitenbucher, J Guy.
Afiliación
  • Gomez L; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Xu R; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Sinko W; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Selfridge B; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Vernier W; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Ly K; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Truong R; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Metz M; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Marrone T; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Sebring K; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Yan Y; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Appleton B; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Aertgeerts K; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Massari ME; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
  • Breitenbucher JG; Dart Neuroscience LLC , 12278 Scripps Summit Drive , San Diego , California 92131 , United States.
J Med Chem ; 61(17): 7754-7766, 2018 09 13.
Article en En | MEDLINE | ID: mdl-30070482

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Conformación Proteica / Quinazolinas / Triazoles / Inhibidores Enzimáticos / Fosfodiesterasas de Nucleótidos Cíclicos Tipo 2 / Modelos Teóricos Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Conformación Proteica / Quinazolinas / Triazoles / Inhibidores Enzimáticos / Fosfodiesterasas de Nucleótidos Cíclicos Tipo 2 / Modelos Teóricos Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Estados Unidos Pais de publicación: Estados Unidos