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Imidazo[2,1-b]benzothiazol Derivatives as Potential Allosteric Inhibitors of the Glucocorticoid Receptor.
Christodoulou, Michael S; Dapiaggi, Federico; Ghiringhelli, Francesca; Pieraccini, Stefano; Sironi, Maurizio; Lucafò, Marianna; Curci, Debora; Decorti, Giuliana; Stocco, Gabriele; Chirumamilla, Chandra Sekhar; Vanden Berghe, Wim; Balaguer, Patrick; Michel, Benoît Y; Burger, Alain; Beccalli, Egle M; Passarella, Daniele; Martinet, Nadine.
Afiliación
  • Christodoulou MS; DISFARM, Sezione di Chimica Generale e Organica "A. Marchesini", Università degli Studi di Milano, Via Venezian 21, 20133 Milano, Italy.
  • Dapiaggi F; Department of Chemistry, Università degli Studi di Milano, Via Golgi 19, 20133 Milano Italy.
  • Ghiringhelli F; Department of Chemistry, Università degli Studi di Milano, Via Golgi 19, 20133 Milano Italy.
  • Pieraccini S; Department of Chemistry, Università degli Studi di Milano, Via Golgi 19, 20133 Milano Italy.
  • Sironi M; Istituto di Scienze e Tecnologie Molecolari (INSTM), CNR, and INSTM, UdR Milano, Via Golgi 19, 20133 Milano, Italy.
  • Lucafò M; Department of Chemistry, Università degli Studi di Milano, Via Golgi 19, 20133 Milano Italy.
  • Curci D; Istituto di Scienze e Tecnologie Molecolari (INSTM), CNR, and INSTM, UdR Milano, Via Golgi 19, 20133 Milano, Italy.
  • Decorti G; Department of Medicine, Surgery and Health Sciences, University of Trieste, 34127 Trieste, Italy.
  • Stocco G; PhD School in Reproduction and Developmental Sciences, University of Trieste, 34127 Trieste, Italy.
  • Chirumamilla CS; Department of Medicine, Surgery and Health Sciences, University of Trieste, 34127 Trieste, Italy.
  • Vanden Berghe W; Institute for Maternal and Child Health - IRCCS "Burlo Garofolo", 34127 Trieste, Italy.
  • Balaguer P; Department of Life Sciences, University of Trieste, 34127 Trieste, Italy.
  • Michel BY; Laboratory of Protein Chemistry, Proteomics and Epigenetic Signalling, Department of Biomedical Sciences, University of Antwerp (UA), 2000 Antwerpen, Belgium.
  • Burger A; Laboratory of Protein Chemistry, Proteomics and Epigenetic Signalling, Department of Biomedical Sciences, University of Antwerp (UA), 2000 Antwerpen, Belgium.
  • Beccalli EM; IRCM, INSERM U1194, Université Montpellier, ICM, 208 rue des Apothicaires, F-34298 Montpellier, France.
  • Passarella D; Université Côte d'Azur, CNRS, Institut de Chimie de Nice, UMR 7272, Parc Valrose, 06108 Nice Cedex 2, France.
  • Martinet N; Université Côte d'Azur, CNRS, Institut de Chimie de Nice, UMR 7272, Parc Valrose, 06108 Nice Cedex 2, France.
ACS Med Chem Lett ; 9(4): 339-344, 2018 Apr 12.
Article en En | MEDLINE | ID: mdl-29670697

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2018 Tipo del documento: Article País de afiliación: Italia Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2018 Tipo del documento: Article País de afiliación: Italia Pais de publicación: Estados Unidos