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Rational Drug Design of Topically Administered Caspase 1 Inhibitors for the Treatment of Inflammatory Acne.
Fournier, Jean-François; Clary, Laurence; Chambon, Sandrine; Dumais, Laurence; Harris, Craig Steven; Millois, Corinne; Pierre, Romain; Talano, Sandrine; Thoreau, Étienne; Aubert, Jérome; Aurelly, Michèle; Bouix-Peter, Claire; Brethon, Anne; Chantalat, Laurent; Christin, Olivier; Comino, Catherine; El-Bazbouz, Ghizlane; Ghilini, Anne-Laurence; Isabet, Tatiana; Lardy, Claude; Luzy, Anne-Pascale; Mathieu, Céline; Mebrouk, Kenny; Orfila, Danielle; Pascau, Jonathan; Reverse, Kevin; Roche, Didier; Rodeschini, Vincent; Hennequin, Laurent François.
Afiliación
  • Fournier JF; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Clary L; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Chambon S; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Dumais L; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Harris CS; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Millois C; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Pierre R; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Talano S; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Thoreau É; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Aubert J; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Aurelly M; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Bouix-Peter C; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Brethon A; Edelris , 115 Avenue Lacassagne , 69003 Lyon , France.
  • Chantalat L; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Christin O; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Comino C; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • El-Bazbouz G; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Ghilini AL; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Isabet T; Synchrotron Soleil , L'Orme des Merisiers, Saint-Aubin, BP 48 , 91192 Gif-sur-Yvette Cedex, France.
  • Lardy C; Edelris , 115 Avenue Lacassagne , 69003 Lyon , France.
  • Luzy AP; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Mathieu C; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Mebrouk K; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Orfila D; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Pascau J; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Reverse K; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
  • Roche D; Edelris , 115 Avenue Lacassagne , 69003 Lyon , France.
  • Rodeschini V; Edelris , 115 Avenue Lacassagne , 69003 Lyon , France.
  • Hennequin LF; Nestlé Skin Health R&D , 2400 Route des Colles, BP 87 , 06902 Sophia-Antipolis Cedex, France.
J Med Chem ; 61(9): 4030-4051, 2018 05 10.
Article en En | MEDLINE | ID: mdl-29648825

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Diseño de Fármacos / Acné Vulgar / Caspasa 1 / Inhibidores de Caspasas Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Francia Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Diseño de Fármacos / Acné Vulgar / Caspasa 1 / Inhibidores de Caspasas Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Francia Pais de publicación: Estados Unidos