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Discovery of selective protein arginine methyltransferase 5 inhibitors and biological evaluations.
Ji, Sen; Ma, Shuang; Wang, Wen-Jing; Huang, Shen-Zhen; Wang, Tian-Qi; Xiang, Rong; Hu, Yi-Guo; Chen, Qiang; Li, Lin-Li; Yang, Sheng-Yong.
Afiliación
  • Ji S; State Key Laboratory of Biotherapy/Collaborative Innovation Center of Biotherapy, West China Hospital, West China Medical School, Sichuan University, Chengdu, Sichuan, China.
  • Ma S; State Key Laboratory of Biotherapy/Collaborative Innovation Center of Biotherapy, West China Hospital, West China Medical School, Sichuan University, Chengdu, Sichuan, China.
  • Wang WJ; State Key Laboratory of Biotherapy/Collaborative Innovation Center of Biotherapy, West China Hospital, West China Medical School, Sichuan University, Chengdu, Sichuan, China.
  • Huang SZ; State Key Laboratory of Biotherapy/Collaborative Innovation Center of Biotherapy, West China Hospital, West China Medical School, Sichuan University, Chengdu, Sichuan, China.
  • Wang TQ; Department of Clinical Medicine, School of Medicine, Nankai University, Tianjin, China.
  • Xiang R; Department of Clinical Medicine, School of Medicine, Nankai University, Tianjin, China.
  • Hu YG; State Key Laboratory of Biotherapy/Collaborative Innovation Center of Biotherapy, West China Hospital, West China Medical School, Sichuan University, Chengdu, Sichuan, China.
  • Chen Q; State Key Laboratory of Biotherapy/Collaborative Innovation Center of Biotherapy, West China Hospital, West China Medical School, Sichuan University, Chengdu, Sichuan, China.
  • Li LL; West China School of Pharmacy, Sichuan University, Chengdu, Sichuan, China.
  • Yang SY; State Key Laboratory of Biotherapy/Collaborative Innovation Center of Biotherapy, West China Hospital, West China Medical School, Sichuan University, Chengdu, Sichuan, China.
Chem Biol Drug Des ; 89(4): 585-598, 2017 04.
Article en En | MEDLINE | ID: mdl-27714957

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Proteína-Arginina N-Metiltransferasas / Inhibidores Enzimáticos Límite: Humans Idioma: En Revista: Chem Biol Drug Des Asunto de la revista: BIOQUIMICA / FARMACIA / FARMACOLOGIA Año: 2017 Tipo del documento: Article País de afiliación: China Pais de publicación: Reino Unido

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Proteína-Arginina N-Metiltransferasas / Inhibidores Enzimáticos Límite: Humans Idioma: En Revista: Chem Biol Drug Des Asunto de la revista: BIOQUIMICA / FARMACIA / FARMACOLOGIA Año: 2017 Tipo del documento: Article País de afiliación: China Pais de publicación: Reino Unido