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TCH1036, a indeno[1,2-c]quinoline derivative, potentially inhibited the growth of human brain malignant glioma (GBM) 8401 cells via suppression of the expression of Suv39h1 and PARP.
Liao, Hsien-Feng; Lee, Chien-Chin; Hsiao, Pei-Chi; Chen, Yi-Fong; Tseng, Chih-Hua; Tzeng, Cherng-Chyi; Chen, Yeh-Long; Chen, Jui-Chang; Chang, Ya-Sian; Chang, Jan-Gowth.
Afiliación
  • Liao HF; The Ph.D. Program for Cancer Biology and Drug Discovery, China Medical University and Academia Sinica, Taichung 40402, Taiwan; School of Medicine, China Medical University, Taichung 40402, Taiwan.
  • Lee CC; Epigenome Research Center, China Medical University Hospital, Taichung 40402, Taiwan.
  • Hsiao PC; Graduate Institute of applied Chemistry, National Chiayi University, Chiayi 60004, Taiwan.
  • Chen YF; The Ph.D. Program for Cancer Biology and Drug Discovery, China Medical University and Academia Sinica, Taichung 40402, Taiwan; School of Medicine, China Medical University, Taichung 40402, Taiwan.
  • Tseng CH; School of Pharmacy, College of Pharmacy, Kaohsiung Medical University, Kaohsiung 80761, Taiwan.
  • Tzeng CC; Department of Medicinal and Applied Chemistry, Kaohsiung Medical University, Kaohsiung 80761, Taiwan.
  • Chen YL; Department of Medicinal and Applied Chemistry, Kaohsiung Medical University, Kaohsiung 80761, Taiwan.
  • Chen JC; Graduate Institute of applied Chemistry, National Chiayi University, Chiayi 60004, Taiwan.
  • Chang YS; Epigenome Research Center, China Medical University Hospital, Taichung 40402, Taiwan; Department of Laboratory Medicine, China Medical University Hospital, Taichung 40402, Taiwan. Electronic address: t25074@mail.cmuh.org.tw.
  • Chang JG; The Ph.D. Program for Cancer Biology and Drug Discovery, China Medical University and Academia Sinica, Taichung 40402, Taiwan; School of Medicine, China Medical University, Taichung 40402, Taiwan; Epigenome Research Center, China Medical University Hospital, Taichung 40402, Taiwan; Department of Lab
Biomed Pharmacother ; 82: 649-59, 2016 Aug.
Article en En | MEDLINE | ID: mdl-27470408

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Oximas / Quinolinas / Proteínas Represoras / Neoplasias Encefálicas / Poli(ADP-Ribosa) Polimerasa-1 / Glioma / Metiltransferasas Límite: Humans Idioma: En Revista: Biomed Pharmacother Año: 2016 Tipo del documento: Article País de afiliación: Taiwán Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Oximas / Quinolinas / Proteínas Represoras / Neoplasias Encefálicas / Poli(ADP-Ribosa) Polimerasa-1 / Glioma / Metiltransferasas Límite: Humans Idioma: En Revista: Biomed Pharmacother Año: 2016 Tipo del documento: Article País de afiliación: Taiwán Pais de publicación: Francia