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Impact of Stepwise NH2-Methylation of Triapine on the Physicochemical Properties, Anticancer Activity, and Resistance Circumvention.
Kowol, Christian R; Miklos, Walter; Pfaff, Sarah; Hager, Sonja; Kallus, Sebastian; Pelivan, Karla; Kubanik, Mario; Enyedy, Éva A; Berger, Walter; Heffeter, Petra; Keppler, Bernhard K.
Afiliación
  • Kowol CR; Institute of Inorganic Chemistry, University of Vienna , Waehringer Str. 42, A-1090 Vienna, Austria.
  • Miklos W; Research Platform "Translational Cancer Therapy Research", University of Vienna , Waehringer Str. 42, A-1090 Vienna, Austria.
  • Pfaff S; Institute of Cancer Research, Medical University of Vienna , Borschkeg. 8a, A-1090 Vienna, Austria.
  • Hager S; Institute of Inorganic Chemistry, University of Vienna , Waehringer Str. 42, A-1090 Vienna, Austria.
  • Kallus S; Institute of Cancer Research, Medical University of Vienna , Borschkeg. 8a, A-1090 Vienna, Austria.
  • Pelivan K; Institute of Inorganic Chemistry, University of Vienna , Waehringer Str. 42, A-1090 Vienna, Austria.
  • Kubanik M; Institute of Inorganic Chemistry, University of Vienna , Waehringer Str. 42, A-1090 Vienna, Austria.
  • Enyedy ÉA; Institute of Inorganic Chemistry, University of Vienna , Waehringer Str. 42, A-1090 Vienna, Austria.
  • Berger W; Department of Inorganic and Analytical Chemistry, University of Szeged , Dóm tér 7, 6720 Szeged, Hungary.
  • Heffeter P; Institute of Cancer Research, Medical University of Vienna , Borschkeg. 8a, A-1090 Vienna, Austria.
  • Keppler BK; Research Platform "Translational Cancer Therapy Research", University of Vienna , Waehringer Str. 42, A-1090 Vienna, Austria.
J Med Chem ; 59(14): 6739-52, 2016 07 28.
Article en En | MEDLINE | ID: mdl-27336684

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piridinas / Tiosemicarbazonas / Antineoplásicos Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2016 Tipo del documento: Article País de afiliación: Austria Pais de publicación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piridinas / Tiosemicarbazonas / Antineoplásicos Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2016 Tipo del documento: Article País de afiliación: Austria Pais de publicación: Estados Unidos