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TRPV1 modulators: Synthesis and in vitro evaluation of 1-heteroaryl piperidinecarboxamide and piperazinylurea derivatives.
Congiu, Cenzo; Onnis, Valentina; Balboni, Gianfranco; Schiano-Moriello, Aniello; Di Marzo, Vincenzo; De Petrocellis, Luciano.
Afiliación
  • Congiu C; Department of Life and Environmental Sciences, Unit of Pharmaceutical, Pharmacological and Nutraceutical Sciences, University of Cagliari, Via Ospedale 72, 09124 Cagliari, Italy. Electronic address: ccongiu@unica.it.
  • Onnis V; Department of Life and Environmental Sciences, Unit of Pharmaceutical, Pharmacological and Nutraceutical Sciences, University of Cagliari, Via Ospedale 72, 09124 Cagliari, Italy.
  • Balboni G; Department of Life and Environmental Sciences, Unit of Pharmaceutical, Pharmacological and Nutraceutical Sciences, University of Cagliari, Via Ospedale 72, 09124 Cagliari, Italy.
  • Schiano-Moriello A; Endocannabinoid Research Group, Institute of Biomolecular Chemistry, National Research Council, Via Campi Flegrei 34, Comprensorio Olivetti, 80078 Pozzuoli, Naples, Italy.
  • Di Marzo V; Endocannabinoid Research Group, Institute of Biomolecular Chemistry, National Research Council, Via Campi Flegrei 34, Comprensorio Olivetti, 80078 Pozzuoli, Naples, Italy.
  • De Petrocellis L; Endocannabinoid Research Group, Institute of Biomolecular Chemistry, National Research Council, Via Campi Flegrei 34, Comprensorio Olivetti, 80078 Pozzuoli, Naples, Italy.
Eur J Med Chem ; 100: 129-38, 2015 Jul 15.
Article en En | MEDLINE | ID: mdl-26079089

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piperidinas / Urea / Canales Catiónicos TRPV / Amidas Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2015 Tipo del documento: Article Pais de publicación: Francia

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Piperidinas / Urea / Canales Catiónicos TRPV / Amidas Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2015 Tipo del documento: Article Pais de publicación: Francia