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Synthesis and biological evaluation of novel selective androgen receptor modulators (SARMs). Part I.
Aikawa, Katsuji; Miyawaki, Toshio; Hitaka, Takenori; Imai, Yumi N; Hara, Takahito; Miyazaki, Junichi; Yamaoka, Masuo; Kusaka, Masami; Kanzaki, Naoyuki; Tasaka, Akihiro; Shiraishi, Mitsuru; Yamamoto, Satoshi.
Afiliación
  • Aikawa K; Pharmaceutical Research Division, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-higashi 2-chome, Fujisawa, Kanagawa 251-85555, Japan. Electronic address: katsuji.aikawa@takeda.com.
  • Miyawaki T; Pharmaceutical Research Division, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-higashi 2-chome, Fujisawa, Kanagawa 251-85555, Japan.
  • Hitaka T; Pharmaceutical Research Division, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-higashi 2-chome, Fujisawa, Kanagawa 251-85555, Japan.
  • Imai YN; Pharmaceutical Research Division, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-higashi 2-chome, Fujisawa, Kanagawa 251-85555, Japan.
  • Hara T; Pharmaceutical Research Division, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-higashi 2-chome, Fujisawa, Kanagawa 251-85555, Japan.
  • Miyazaki J; Pharmaceutical Production Division, Takeda Pharmaceutical Company Ltd, 17-85 Jusohommachi 2-chome, Yodogawa-ku, Osaka 532-8686, Japan.
  • Yamaoka M; Pharmaceutical Research Division, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-higashi 2-chome, Fujisawa, Kanagawa 251-85555, Japan.
  • Kusaka M; CMC Center, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-higashi 2-chome, Fujisawa, Kanagawa 251-85555, Japan.
  • Kanzaki N; Pharmaceutical Research Division, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-higashi 2-chome, Fujisawa, Kanagawa 251-85555, Japan.
  • Tasaka A; Environment & Safety Department, Takeda Pharmaceutical Company Ltd, 17-85 Jusohommachi 2-chome, Yodogawa-ku, Osaka 532-8686, Japan.
  • Shiraishi M; Laboratories of Medicinal & Organic Chemistry Pharmaceutical Sciences, Himeji Dokkyo University, 7-2-1, Kamiohno, Himeji-shi, Hyogo 670-8524, Japan.
  • Yamamoto S; Pharmaceutical Research Division, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-higashi 2-chome, Fujisawa, Kanagawa 251-85555, Japan.
Bioorg Med Chem ; 23(10): 2568-78, 2015 May 15.
Article en En | MEDLINE | ID: mdl-25862209

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pirrolidinas / Receptores Androgénicos / Anabolizantes / Andrógenos / Naftoles Límite: Animals / Humans / Male Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2015 Tipo del documento: Article Pais de publicación: Reino Unido

Texto completo: 1 Colección: 01-internacional Base de datos: MEDLINE Asunto principal: Pirrolidinas / Receptores Androgénicos / Anabolizantes / Andrógenos / Naftoles Límite: Animals / Humans / Male Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2015 Tipo del documento: Article Pais de publicación: Reino Unido