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Parasitol Res ; 114(4): 1313-26, 2015 Apr.
Artículo en Inglés | MEDLINE | ID: mdl-25566774

RESUMEN

Chagas disease, caused by the protozoan Trypanosoma cruzi, is a major parasitic disease that affects millions of people in America. However, despite the high impact of this disease on human health, no effective and safe treatment has been found that eliminates the infecting parasite from human patients. Among the possible chemotherapeutic targets that could be considered for study in T. cruzi are the DNA polymerases, in particular DNA polymerase beta (polß), which previous studies have shown to be involved in kinetoplast DNA replication and repair. In this paper, we describe the expression, purification, and biochemical characterization of the Miranda clone polß, corresponding to lineage T. cruzi I (TcI). The recombinant enzyme purified to homogeneity displayed specific activity in the range described for a highly purified mammalian polß. However, the trypanosome enzyme exhibited important differences in biochemical properties compared to the mammalian enzymes, specifically an almost absolute dependency on KCl, high sensitivity to N-ethylmaleimide (NEM), and low sensitivity to ddTTP. Immuno-affinity purification of T. cruzi polymerase beta (Tcpolß) from epimastigote extracts showed that the native enzyme was phosphorylated. In addition, it was demonstrated that Tcpolß interacts with some proteins in a group of about 15 proteins which are required to repair 1-6 bases of gaps of a double strand damaged DNA. It is possible that these proteins form part of a DNA repair complex, analogous to that described in mammals and some trypanosomatids.


Asunto(s)
Enfermedad de Chagas/parasitología , ADN Polimerasa beta/genética , Regulación Enzimológica de la Expresión Génica , Trypanosoma cruzi/enzimología , ADN Polimerasa beta/efectos de los fármacos , ADN Polimerasa beta/aislamiento & purificación , ADN Polimerasa beta/metabolismo , ADN de Cinetoplasto/química , ADN de Cinetoplasto/genética , Didesoxinucleótidos/farmacología , Inhibidores Enzimáticos/farmacología , Escherichia coli/genética , Escherichia coli/metabolismo , Etilmaleimida/farmacología , Humanos , Fosforilación , Filogenia , Análisis de Secuencia de ADN , Nucleótidos de Timina/farmacología , Trypanosoma cruzi/genética
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