1.
Org Biomol Chem
; 19(43): 9514, 2021 Nov 10.
Artículo
en Inglés
| MEDLINE
| ID: mdl-34709276
RESUMEN
Correction for 'I2/TBHP mediated diastereoselective synthesis of spiroaziridines' by Kizhakkan Thiruthi Ashitha et al., Org. Biomol. Chem., 2020, 18, 1588-1593, DOI: 10.1039/C9OB02711D.
2.
Org Biomol Chem
; 18(8): 1588-1593, 2020 02 26.
Artículo
en Inglés
| MEDLINE
| ID: mdl-32048676
RESUMEN
Eventhough spiroheterocycles are considered as emerging drug candidates, synthesis of spiroaziridines has not been well explored so far. Herein, we disclose an efficient I2/TBHP mediated diastereoselective synthesis of N-alkyl spiroaziridines from primary amines and easily accessible α,ß-unsaturated ketones. The reaction is also compatible for the synthesis of 2-aroylaziridines.