1.
Bioorg Med Chem Lett
; 18(18): 5087-90, 2008 Sep 15.
Artículo
en Inglés
| MEDLINE
| ID: mdl-18752951
RESUMEN
A novel series of bacterial topoisomerase (3-aminoquinazolinediones) inhibitors are described. The side-chain SAR against Gram-positive and Gram-negative organisms as well as DNA gyrase activity is reported.