1.
Chem Commun (Camb)
; 57(19): 2388-2391, 2021 Mar 07.
Artículo
en Inglés
| MEDLINE
| ID: mdl-33538721
RESUMEN
In an effort designed to discover superior inhibitors of cyclophilin D (CypD), we identified and screened members of a one-bead-one-compound (OBOC) library of cyclic peptoid analogues of cyclosporin A (CsA). The results show that the one member of this cyclic peptoid family, I11, inhibits mitochondrial membrane potential changes mediated by CypD.