1.
Bioorg Med Chem
; 13(22): 6218-25, 2005 Nov 15.
Artículo
en Inglés
| MEDLINE
| ID: mdl-16061385
RESUMEN
A series of C-4-anilino- and C-4-imido-substituted new podophyllotoxin congeners have been designed, synthesized, and evaluated for their cytotoxicity and DNA topoisomerase-II (topo-II) inhibition potential. Some of these compounds have exhibited promising in vitro anticancer and topo-II inhibition activity.