1.
Bioorg Med Chem Lett
; 16(1): 186-90, 2006 Jan 01.
Artículo
en Inglés
| MEDLINE
| ID: mdl-16260134
RESUMEN
As part of a detailed study, the syntheses, biological activities, and pharmacokinetic properties of hydroxylated analogues of the previously described broad spectrum antifungal agents, Sch 51048 (1), Sch 50001 (3), and Sch 50002 (4), are described. Based on an overall superior profile, one of the alcohols, Sch 56592 (2), was selected for clinical studies.