1.
Bioorg Med Chem Lett
; 17(20): 5537-42, 2007 Oct 15.
Artículo
en Inglés
| MEDLINE
| ID: mdl-17766107
RESUMEN
A novel potent NMDA-NR2B selective antagonist without the reactive metabolites formation issue was identified. Through this study, a close correlation between reactive metabolites formation and calculated HOMO energies of parent compounds was found.