1.
Biosci Biotechnol Biochem
; 68(10): 2178-82, 2004 Oct.
Artículo
en Inglés
| MEDLINE
| ID: mdl-15502365
RESUMEN
The structure-activity relationship for FR901464, a potent cell-cycle inhibitor, was examined by synthesizing its analogs. A versatile method for converting FR901464 was devised. This method made it possible to synthesize biologically active FR901464-biotin conjugates which could be used to isolate the binding proteins.