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Phytochemistry ; 71(8-9): 964-74, 2010 Jun.
Artículo en Inglés | MEDLINE | ID: mdl-20356612

RESUMEN

In an effort to find antimalarial drugs, a systematic in vitro evaluation on a chloroquine-resistant strain of Plasmodium falciparum (FcB1) was undertaken on sixty plant extracts collected in French Guiana. The ethyl acetate extract obtained from the root barks of Symphonia globulifera exhibited a strong antiplasmodial activity (97% at 10 microg/ml). The phytochemical investigation of this extract led to the isolation of nine polycyclic polyprenylated acylphloroglucinol (PPAPs) compounds and two oxidized derivatives. All compounds showed antiplasmodial activity with IC(50)s ranged from 2.1 to 10.1 microM. A LC/ESI-MS(n) study performed on polyprenylated benzophenones previously isolated from Moronobea coccinea provided a reliable method for their detection in the extract and structural elucidation.


Asunto(s)
Antimaláricos/aislamiento & purificación , Antimaláricos/farmacología , Benzofenonas/aislamiento & purificación , Benzofenonas/farmacología , Clusiaceae/química , Plasmodium falciparum/efectos de los fármacos , Antimaláricos/química , Benzofenonas/química , Cloroquina/farmacología , Resistencia a Medicamentos/efectos de los fármacos , Fibroblastos/efectos de los fármacos , Guyana Francesa , Humanos , Estructura Molecular , Resonancia Magnética Nuclear Biomolecular , Pruebas de Sensibilidad Parasitaria , Corteza de la Planta/química , Raíces de Plantas/química
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