1.
Bioorg Med Chem Lett
; 10(16): 1803-6, 2000 Aug 21.
Artículo
en Inglés
| MEDLINE
| ID: mdl-10969972
RESUMEN
A weak HTS hit at the CCR2B receptor has been converted into a potent antagonist by array SAR studies. Selectivity over the closely related CCR5 receptor is also achieved.